Course Program

 

  • Introduction, principles and history of Combinatorial Chemistry
  • Methods and Techniques in Combi Chem
  • Characterizations of combinatorial library
  • Overview on the use of combi chem in medicinal chemistry
  • Critics and perspective to combi chem
  • Examples of combi chem in medicinal chemistry
  • Automation and data processing
  • Multicomponent reactions (Biginelli, Passerini, Ugi etc.)
  • Tandem-domino reactions
  • Bioconjugation methods
  • Bioorthogonal reactions
  • Non-covalent bioconjugation strategies 

 

  • Dynamic Combinatorial Chemistry, introduction, history and perspective
  • Exchange reactions
  • Developing of synthetic receptors using DCLs
  • Ligands for Biomolecules
  • Polymers formed by DCC

 

  • Systems chemistry
  • Erwin Schrödinger’s most famous question, what is life?
  • Prebiotic Chemistry. Molecular network interactions and equilibrium
  • Asymmetric synthesis in enantioselective autocatalytic reactions
  • Speculations on chemical evolution. DNA and RNA in chemical evolvable systems
  • The role of amphiphilic interactions on the formation of supramolecular structures